Sustained occupation of pituitary GnRH receptors by Leuprorelin results in desensitization and/or downregulation of receptors in the anterior pituitary, thereby suppressing gonadotrophin release and reducing testosterone release by the human testes to castrate levels.
LORELIN DEPOT INJ. 3.75MG/7.5MG/11.25MG
Generic Name: Leuprorelin Acetate
Indications
Leuprorelin Acetate is used for treating prostatic cancer, endometriosis, premenopausal breast cancer, uterine myoma, and central precocious puberty.
It also helps manage PCOS, severe PMS, and functional bowel disease, and is being investigated for Alzheimer’s disease.